Observed performance metrics in laboratory models
Observed performance metrics in laboratory models
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Research summary on Cardarine (also known as GW-501506).
It’s technically not a SARM — but it’s often grouped with them because of how it's used.
Cardarine is a PPAR delta agonist — which means it activates pathways in the tissue that turn stored fat into usable energy.
In research settings, Cardarine has been shown to:
✔ Increase respiratory oxygenation in lung tissue.
✔ Enhance fatty acid transport and oxidation.
✔ And support metabolic function — especially in skeletal muscle and cardiac tissue.
🔥 CARDIAC ENDURANCE:
In studies, Cardarine has shown to increase oxygen utilization in lung tissue — helping muscle tissue operate under higher workloads without depleting glycogen stores as rapidly.
🫓 FAT OXIDATION:
Cardarine activates genes involved in the fatty acid transport process. Additionally, it enhances intracellular fatty acid transport and oxidation, leading to more efficient energy utilization in muscle tissue.
⚡️ MUSCULAR ENDURANCE:
Cardarine enhances how efficiently cells produce energy — especially in skeletal muscle and heart tissue — allowing those systems to operate longer without fatiguing as quickly.
1. PPAR Promotes Running Endurance by Preserving Glucose
https://www.cell.com/cell-metabolism/pdf/S1550-4131%2817%2930211-5.pdf
2. A metabolomic study of the PPAR agonist GW501516 for enhancing running endurance in Kunming mice
https://www.nature.com/articles/srep09884
3. Cardarine (GW501516) Effects on Improving Metabolic Syndrome
4. GW501516 (Cardarine): Pharmacological and Clinical Effects
https://www.scivisionpub.com/pdfs/gw501516-cardarine-pharmacological-and-clinical-effects-2879.pdf
5. Activation of PPAR signaling improves skeletal muscle oxidative metabolism
https://pmc.ncbi.nlm.nih.gov/articles/PMC4551122/
6. PPAR-agonist GW501516 ameliorates insulin resistance in mice
https://pubmed.ncbi.nlm.nih.gov/18684227/
7. Lipid effects of GW501516 in dyslipidemic subjects
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